Search
Titanium Dioxide Acetic Acid Citric Acid Sodium Hydroxide Oxalic Acid Ethyl Acetate
Sign in/Join free

Product Details & Description

Product Info
Product Name Tirzepatide
CAS No. 2023788-19-2
Catalog No. HH482502737210201699
Brand Hebei saisier
Purity -
Packing -
Package -
Lead Time -
Origin -
Loading Port -
Chemical Identifiers
Melting Point -
Boiling Point -
Water Solubility -
Density -
Storage Temp Store at -20°C
Flash Point -
Stability -
Appearance White to off-white Solid
Refractive Index -
Product Info

抗糖尿病药物替西帕肽是胰高血糖素样肽-1受体(GLP-1)和葡萄糖依赖性促胰岛素多肽(GIP,也称为胃抑制性多肽)的新型双重激动剂,每周给药一次。GLP-1 和 GIP 都是肠促胰岛素,是人体胃肠道粘膜分泌的肽。Tirzepatide 与胰岛细胞上的受体结合并刺激胰岛素分泌,从而降低血糖。它还可以延迟胃排空并抑制食欲,从而控制体重。而替西帕肽则抑制胃酸和胃蛋白酶分泌,刺激胰岛素释放,抑制胃蠕动和排空,补充GLP-1受体激动剂的作用。Tirzepatide 将两种促胰岛素作用整合到一个分子中,代表了一类治疗 2 型糖尿病的新型药物。


Tirzepatide 与索马鲁肽具有相似的序列。序列中的 Lys 侧链用 PEG 修饰,PEG 是一种在肽中发现的官能团,已知可增加水溶性。Tirzepatide的主要生理功能是葡萄糖依赖性胰岛素多肽(GIP)和胰高血糖素样肽-1(GLP-1)受体的双重激动剂。它正在开发用于治疗 2 型糖尿病,并已进入临床阶段。

Request For Quotation

Tirzepatide

2023788-19-2

Other Supplier Reference

Product name
Purity
Packing
Lead Time
Country
Company Name
Details
0.99
GlassBottle kg
China
Request For Quotation
99.99%
5mg 10mg 15mg 20mg 30mg 40mg 50mg 60mg
China
Request For Quotation
99%
1g/bottle
China
Request For Quotation
99%
G/KG
China
Request For Quotation
99%
1kg/bag,25kg/drum,25kg/bag
China
Request For Quotation
99%
1kg/bag;25kg/Cardboard Drum
China
Request For Quotation
99%
5mg/10mg/15mg per vial; 1g,10g or according to customer's detail requirement.
China
Request For Quotation
99%
10mg/vial,10vials/box
China
Request For Quotation
99%
bag/mg
China
Request For Quotation